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The Mitomycin Antibiotics. Synthetic Studies. XV.1 The Preparation of a Related Indoloquinone2 George R. Allen and Martin J. Weiss pp 1 - 6; DOI: 10.1021/jm00313a001 |
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The Mitomycin Antibiotics. Synthetic Studies. XVI.1 The Utilization of 5-Methoxy-4-nitro-3-indolecarboxaldehydes for the Synthesis of Related 4,7-Indoloquinones2 George R. Allen, Louis J. Binovi, and Martin J. Weiss pp 7 - 13; DOI: 10.1021/jm00313a002 |
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The Mitomycin Antibiotics. Synthetic Studies. XVII.1 Indoloquinone Analogs with Variants at the 2 Position George R. Allen, John F. Poletto, and Martin J. Weiss pp 14 - 22; DOI: 10.1021/jm00313a003 |
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The Mitomycin Antibiotics. Synthetic Studies. XVIII.1 Preparation of 1-(β-Substituted ethyl)indoloquinone Analogs George R. Allen and Martin J. Weiss pp 23 - 29; DOI: 10.1021/jm00313a004 |
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Antimicrobial Properties of Pyrrole Derivatives Albert J. Castro, Glen R. Gale, Gary E. Means, and Gerard Tertzakian pp 29 - 32; DOI: 10.1021/jm00313a005 |
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Organophosphorus Compounds as Schistosomicides Leslie M. Werbel and Paul E. Thompson pp 32 - 36; DOI: 10.1021/jm00313a006 |
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Mixed Bifunctionality. Antitumor Properties of 2-Chloroethyl Sulfide Derivatives of Polynuclear Aromatic Hydrocarbons Richard M. Peck, Anna P. O'Connell, and Hugh J. Creech pp 37 - 40; DOI: 10.1021/jm00313a007 |
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Acetylenic Carbamates. A New Class of Potential Oncolytic Agents Robert D. Dillard, Gerald Poore, Donald R. Cassady, and Nelson R. Easton pp 40 - 44; DOI: 10.1021/jm00313a008 |
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The 6-Deoxytetracyclines. VII. Alkylated Aminotetracyclines Possessing Unique Antibacterial Activity Michael J. Martell and James H. Boothe pp 44 - 46; DOI: 10.1021/jm00313a009 |
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Nucleosides. XXXVII. 5,6-Substituted 5-Fluorodihydropyrimidines and Their 2′-Deoxyribonucleosides R. Duschinsky, T. Gabriel, W. Tautz, A. Nussbaum, M. Hoffer, E. Grunberg, J. H. Burchenal, and J. J. Fox pp 47 - 58; DOI: 10.1021/jm00313a010 |
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Irreversible Enzyme Inhibitors. LXXIII.1,2 Inhibitors of Guanine Deaminase. I. Mode of Binding of Guanine B. R. Baker pp 59 - 61; DOI: 10.1021/jm00313a011 |
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Irreversible Enzyme Inhibitors. LXXIV. Inhibitors of Guanine Deaminase. II. Studies on Bulk Tolerance within Enzyme-Inhibitor Complexes B. R. Baker and Daniel V. Santi pp 62 - 64; DOI: 10.1021/jm00313a012 |
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Experimentally Induced Phenylketonuria. I. Inhibitors of Phenylalanine Hydroxylase Joseph I. DeGraw, Michael Cory, W. A. Skinner, Myna C. Theisen, and Chozo Mitoma pp 64 - 66; DOI: 10.1021/jm00313a013 |
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Pyrazine Diuretics. II. N-Amidino-3-amino-5-substituted 6-Halopyrazinecarboxamides Edward J. Cragoe, Otto W. Woltersdorf, John B. Bicking, Sara F. Kwong, and James H. Jones pp 66 - 75; DOI: 10.1021/jm00313a014 |
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The Effect of Piperidinecarboxamide Derivatives on Isolated Human Plasma Cholinesterase. III. Variation in the N1-Hydrocarbon Substituent James G. Beasley and Linda L. Williford pp 76 - 78; DOI: 10.1021/jm00313a015 |
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Mammalian Antifertility Agents. IV. Basic 3,4-Dihydronaphthalenes and 1,2,3,4-Tetrahydro-1-naphthols Daniel Lednicer, Stanley C. Lyster, and Gordon W. Duncan pp 78 - 84; DOI: 10.1021/jm00313a016 |
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Substituted Aminoalkoxytriarylhaloethylenes Frank P. Palopoli, Vernon J. Feil, Robert E. Allen, Dorsey E. Holtkamp, and Alfred Richardson pp 84 - 86; DOI: 10.1021/jm00313a017 |
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Synthesis and Pharmacological Properties of New 9,10-Dihydro-9,10-ethanoanthracene Derivatives Jacques R. Boissier, Roger Ratouis, Claude Dumont, Laurent Taliani, and Jeannine Forest pp 86 - 91; DOI: 10.1021/jm00313a018 |
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Nitrofuryl Heterocycles. V.1 4-Acyl-5,5-dialkyl-2-(5-nitro-2-furyl)-Δ2-1,3,4-oxadiazolines Homer A. Burch pp 91 - 93; DOI: 10.1021/jm00313a019 |
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Synthesis and Bacteriostatic Activity of Some Nitrotrifluoro methylanilides Joseph W. Baker, Gerald L. Bachman, Ignatius Schumacher, Daniel P. Roman, and Alan L. Tharp pp 93 - 95; DOI: 10.1021/jm00313a020 |
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The Mitomycin Antibiotics. Synthetic Studies. XIX.1 Synthesis of Indoloquinone Analogs with Certain C-3 Variants John F. Poletto, George R. Allen, and Martin J. Weiss pp 95 - 97; DOI: 10.1021/jm00313a021 |
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A Polymeric Nitrofuran Derivative with Prolonged Antibacterial Action Franca Ascoli, Giovanni Casini, Marcello Ferappi, and Ezio Tubaro pp 97 - 99; DOI: 10.1021/jm00313a022 |
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Fluorene Derivatives for Antitumor Activity Krishna C. Agrawal pp 99 - 101; DOI: 10.1021/jm00313a023 |
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New Alkylating Agents Derived from Diaziridine Csaba Szantay, Z. F. Chmielewicz, and T. J. Bardos pp 101 - 104; DOI: 10.1021/jm00313a024 |
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Aminomethylation and Hydroxymethylation of Purine-6(1H)-thione and 6-Alkylthiopurines C. P. Bryant and R. E. Harmon pp 104 - 106; DOI: 10.1021/jm00313a025 |
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The Preparation of α-Phenylketo Steroids John F. Poletto, George R. Allen, and Martin J. Weiss pp 106 - 108; DOI: 10.1021/jm00313a026 |
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Isobutyl N-Chloroethyl-N-nitrosocarbamate W. C. J. Ross pp 108 - 109; DOI: 10.1021/jm00313a027 |
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Abolition of Immunosuppressive Activity of 6-Mercaptopurine and Thioguanine by 8-Phenyl Substitution S.-C. J. Fu, B. J. Hargis, E. Chinoporos, and S. Malkiel pp 109 - 110; DOI: 10.1021/jm00313a028 |
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Heterocycles Containing (8-Hydroxy-5-methyl-7-quinolyl)vinyl Groups Al G. Mueller and J. P. Phillips pp 110 - 111; DOI: 10.1021/jm00313a029 |
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The Photosensitizing Activity of N,N′-Bis(p-formylphenyl)piperazine S. N. Thampi, F. W. Schueler, Vernon B. Haarstad, and Silas E. O'Quinn pp 111 - 112; DOI: 10.1021/jm00313a030 |
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Pyrimidines. V. Some Higher 5-Substituted 2,4,6-Trichloropyrimidines Herman Gershon, Raulo Parmegiani, and Richard D'Ascoli pp 113 - 115; DOI: 10.1021/jm00313a031 |
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Selenophosphorus Compounds as Powerful Cholinesterase Inhibitors Stig Åkerfeldt and Lars Fagerlind pp 115 - 116; DOI: 10.1021/jm00313a032 |
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Phosphorus Analogs of Sulfonylureas. Sodium N-Carbamoylphosphonamidates William J. Fanshawe, Victor J. Bauer, and S. R. Safir pp 116 - 117; DOI: 10.1021/jm00313a033 |
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Pantothenic Acid Derivatives Richard H. Wiley and John E. Kennedy pp 117 - 118; DOI: 10.1021/jm00313a034 |
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Insect Chemosterilants. IV. Phosphoramides Paul H. Terry and Alexej B. Bořkovec pp 118 - 119; DOI: 10.1021/jm00313a035 |
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Effect of Organic Compounds on Reproductive Processes. V. Alkylating Agents Derived from Aryl-, Aralkyl-, and Cyclohexylmethylenediamines W. A. Skinner, M. Cory, T. E. Shellenberger, and J. I. DeGraw pp 120 - 121; DOI: 10.1021/jm00313a036 |
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Structure and Anticoagulant Activity of Bridge-Substituted Dicoumarols R. B. Arora, N. R. Krishnaswamy, T. R. Seshadri, S. D. S. Seth, and B. R. Sharma pp 121 - 124; DOI: 10.1021/jm00313a037 |
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Leguminosae Alkaloids. II. Alkaloids of Lupinus westianus Small Stanley I. Goldberg and Muhammad S. Sahli pp 124 - 125; DOI: 10.1021/jm00313a038 |
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Some Pyrido[2,3-d]thiazole Systems Charles O. Okafor pp 126 - 126; DOI: 10.1021/jm00313a039 |
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Synthesis of the Isoellipticine, 5,11-Dimethyl-10H-pyrido[3,4-b]carbazole Allan N. Fujiwara, Edward M. Acton, and Leon Goodman pp 126 - 127; DOI: 10.1021/jm00313a040 |
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Substituted 1,2,3,4-Tetrahydro-β-carbolines. II J. I. DeGraw, J. G. Kennedy, and W. A. Skinner pp 127 - 128; DOI: 10.1021/jm00313a041 |
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Some Reactions with 4-Cyano-4-phenyltetrahydropyran P. J. Hattersley and I. M. Lockhart pp 128 - 129; DOI: 10.1021/jm00313a042 |
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Vitamin B6 Analogs. An Improved Synthesis of 5-Deoxypyridoxal Peter F. Mühlradt and Esmond E. Snell pp 129 - 130; DOI: 10.1021/jm00313a043 |
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N-Oxides of 9-(β-D-Xylofuranosyl)adenine and 9-(β-D-Arabinofuranosyl)adenine Elmer J. Reist, Dianne F. Calkins, and Leon Goodman pp 130 - 130; DOI: 10.1021/jm00313a044 |
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Esters and Amides from Mannich Ketones G. P. Ellis and T. B. Lee pp 130 - 131; DOI: 10.1021/jm00313a045 |
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Method of Biochemical Analysis. Volume XIV. W. W. Harrison pp 132 - 132; DOI: 10.1021/jm00313a046 |
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Control of Energy Metabolism. William R. Nes pp 132 - 132; DOI: 10.1021/jm00313a047 |
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Synthesis of Some New 17-Spiro-Substituted Steroids Duane F. Morrow, Ruthann M. Hofer, and Townley P. Culbertson pp 133 - 138; DOI: 10.1021/jm00314a001 |
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Synthetic Estrogens, Implantation Inhibitors, and Hypocholesterolemic Agents. I. Tetrahydronaphthalene Series W. L. Bencze, L. I. Barsky, R. W. J. Carney, A. A. Renzi, and George deStevens pp 138 - 144; DOI: 10.1021/jm00314a002 |
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Synthesis of 3β-Acetoxy-17β-(L-arginyl-L-arginyl-L -prolyl)amino-5α-androstane George R. Pettit, Robert L. Smith, and H. Klinger pp 145 - 148; DOI: 10.1021/jm00314a003 |
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Heterocyclic Tetrazoles, a New Class of Lipolysis Inhibitors Gerald F. Holland and Joseph N. Pereira pp 149 - 154; DOI: 10.1021/jm00314a004 |
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The Antifertility Activity of Isoflavones Related to Genistein G. W. Moersch, D. F. Morrow, and W. A. Neuklis pp 154 - 158; DOI: 10.1021/jm00314a005 |
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Cholesterol-Solubilizing Agents Related to the Gallstone Problem C. Ainsworth, D. N. Benslay, J. Davenport, J. L. Hudson, D. Kau, T. M. Lin, and R. R. Pfeiffer pp 158 - 161; DOI: 10.1021/jm00314a006 |
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Synthesis and Some Toxicity and Oxidation Studies of a Fatty Acid Hydroquinone and Analogs of Tocol and δ-Tocopherol Robert A. Stein pp 162 - 164; DOI: 10.1021/jm00314a007 |
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Pteridinecarboxamide Diuretics. II. Reaction of 4,6-Diamino-5-nitrosopyrimidines with N-Substituted Cyanoacetamides T. S. Osdene, Arthur A. Santilli, Lee E. McCardle, and Marvin E. Rosenthale pp 165 - 171; DOI: 10.1021/jm00314a008 |
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Potential Anticancer Agents. II. Urethan-Type Nitrogen Mustards of Some Natural Sex Hormones I. Niculescu-Duvaz, A. Cambanis, and E. Tárnáuceanu pp 172 - 174; DOI: 10.1021/jm00314a009 |
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Histamine Releasers. III. Dibasic Acid Amides of 4-Phenyl-4-aminomethylpiperidines Joseph I. DeGraw, Vernon H. Brown, Nicholas E. Kontaxis, Samuel A. Ferguson, Gale R. Gordon, John H. Peters, and W. A. Skinner pp 174 - 177; DOI: 10.1021/jm00314a010 |
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16-Aza Steroids R. W. Kierstead, A. Faraone, and A. Boris pp 177 - 181; DOI: 10.1021/jm00314a011 |
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Enzyme Inhibitors. XV. A New Irreversible Inhibitor of Adenosine Deaminase Howard J. Schaeffer and Eugene Odin pp 181 - 185; DOI: 10.1021/jm00314a012 |
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Organic Fluorine Compounds. II. Synthesis and Antifungal Properties of 2-Fluoro Fatty Acids Herman Gershon and Raulo Parmegiani pp 186 - 188; DOI: 10.1021/jm00314a013 |
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The Adamantyl Group in Medicinal Agents. III. Nucleoside 5′-Adamantoates. The Adamantoyl Function as a Protecting Group Koert Gerzon and Don Kau pp 189 - 199; DOI: 10.1021/jm00314a014 |
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Totally Synthetic Steroid Hormones. XIII.1 The Chemical Resolution of Some Racemic Estrane, 13β-Ethylgonane, and 13β-n-Propylgonane Derivatives and the Preparation of Some Estrane and 13β-Ethylgonane Derivatives of Unnatural Configuration G. C. Buzby, D. Hartley, G. A. Hughes, Herchel Smith, B. W. Gadsby, and A. B. A. Jansen pp 199 - 204; DOI: 10.1021/jm00314a015 |
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Modification of the Side Chain of Fusidie Acid (Ramycin) G. Janssen and H. Vanderhaeghe pp 205 - 208; DOI: 10.1021/jm00314a016 |
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Anthelmintic Activity of 1,2,4-Oxadiazoles C. Ainsworth, W. E. Buting, J. Davenport, M. E. Callender, and M. C. McCowen pp 208 - 211; DOI: 10.1021/jm00314a017 |
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Derivatives of 1-Hydroxybenzimidazoles and 1-Hydroxyindoles and Their Central Depressant Effects George deStevens, Ann Brooker Brown, David Rose, Harvey I. Chernov, and A. J. Plummer pp 211 - 214; DOI: 10.1021/jm00314a018 |
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A Series of Central Nervous System Stimulants Based on the 4-Substituted 3,3-Diphenyl-2-pyrrolidinone Skeleton. II Albert D. Cale, Herndon Jenkins, Bernard V. Franko, John W. Ward, and Carl D. Lunsford pp 214 - 222; DOI: 10.1021/jm00314a019 |
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1,2-Benzothiazines. IV.1 The Synthesis of 7,8-Dihydropyrido[1,2-b][1,2]benzothiazine-10,11(9H,10aH)-dione 5,5-Dioxides as 1,2-Benzothiazine Analogs of Partial Tetracycline Structures Harold Zinnes, Roger A. Comes, and John Shavel pp 223 - 227; DOI: 10.1021/jm00314a020 |
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1,4,5,6-Tetrahydro-as-triazines. II. Condensation of β-Aminoalkylhydrazines with Iminoesters and Orthoesters Donald L. Trepanier, Jack E. Richman, and Allan D. Rudzik pp 228 - 231; DOI: 10.1021/jm00314a021 |
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The Synthesis and Pharmacology of 131I-Labeled 1,10-Bis(trimethylammonium)-5-chloro-6-iodo-5-decene Dihalide and Related Neuromuscular Blocking Agents Ove A. Nedergaard and Dermot B. Taylor pp 231 - 235; DOI: 10.1021/jm00314a022 |
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The Synthesis and Evaluation of the Local Anesthetic Activity of a Series of 4-(ω-Alkylaminoacylamino)salicylate Esters George Tsatsas, Constantinos Sandris, Demetrios Kontonassios, John F. Zaroslinski, Ronald K. Browne, and Leroy H. Possley pp 235 - 242; DOI: 10.1021/jm00314a023 |
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6-Glycine-8-phenyllactic Acid Bradykinin. Its Synthesis, Biological Activity, and Splitting by Kininase (Carboxypeptidase N) G. A. Ravdel, M. P. Filatova, L. A. Shchukina, T. S. Paskhina, M. S. Surovikina, S. S. Trapeznikova, and T. P. Egorova pp 242 - 246; DOI: 10.1021/jm00314a024 |
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Nucleosides. XXXV. 1-β-D-Arabinofuranosyl-5-methylcytosine Iris L. Doerr, John F. Codington, and Jack J. Fox pp 247 - 248; DOI: 10.1021/jm00314a025 |
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Synthesis of Some Orotic Acid Analogs as Potential Antimetabolites Saul Borodkin, Sigurdur Jonsson, George H. Cocolas, and Robert L. McKee pp 248 - 251; DOI: 10.1021/jm00314a026 |
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Synthesis of a Nonapeptide Sequence of Chymotrypsin T. Mizoguchi and D. W. Woolley pp 251 - 252; DOI: 10.1021/jm00314a027 |
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The Synthesis of the 2α-Methylthio Derivatives of Cortisone, Hydrocortisone, and Progesterone. The Reaction of Methanesulfenyl Chloride with Alkoxalylated Steroid Ketones Henry M. Kissman, Robert E. Schaub, and Martin J. Weiss pp 252 - 254; DOI: 10.1021/jm00314a028 |
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Steroidal γ-Lactones. The Claisen Condensation of 17α-Acetate with 17β-Acetyl G. W. Moersch, D. E. Evans, and G. S. Lewis pp 254 - 255; DOI: 10.1021/jm00314a029 |
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The Synthesis of Some Aryl Nitrogen Mustard Derivatives of Estrogens C. R. Walk, T. C. Chou, and Hsi Hu Lin pp 255 - 257; DOI: 10.1021/jm00314a030 |
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Some Alkylating Derivatives of Nicotinic Acid. Synthesis and Antineoplastic Activities W. C. J. Ross pp 257 - 259; DOI: 10.1021/jm00314a031 |
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Alkylating Activity of 1,3-Bis(2-chloroethyl)-1-nitrosourea and Related Compounds Glynn P. Wheeler and Sue Chumley pp 259 - 261; DOI: 10.1021/jm00314a032 |
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Synthesis of Vitamin B6. III. 3-Deoxypyridoxine Stanton A. Harris, Elbert E. Harris, Elwood R. Peterson, and Edward F. Rogers pp 261 - 262; DOI: 10.1021/jm00314a033 |
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Cyclohexyl Derivatives of Dopacetamide and Dopamine John T. Suh, Claude I. Judd, and Frank E. Kaminski pp 262 - 264; DOI: 10.1021/jm00314a034 |
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Isomeric Mannich Bases Derived from Ethyl 5-Hydroxy-2-methylindole-3-carboxylate M. R. Bell, R. Oesterlin, A. L. Beyler, H. R. Harding, and G. O. Potts pp 264 - 266; DOI: 10.1021/jm00314a035 |
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β-Phenoxyethylamines with Local Anesthetic and Antispasmodic Activity Paolo Da Re, Lucia Verlicchi, and Ivo Setnikar pp 266 - 270; DOI: 10.1021/jm00314a036 |
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The Sulfur Analog of Serotonin E. Campaigne, T. Bosin, and E. S. Neiss pp 270 - 271; DOI: 10.1021/jm00314a037 |
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Some p-Hydroxyphenoxyacetic Acid Derivatives Hikmat T. Fikrat and Nicolas Zenker pp 271 - 273; DOI: 10.1021/jm00314a038 |
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Phosphinylguanidines. Phosphorus Analogs of Biguanides William J. Fanshawe and Victor J. Bauer pp 273 - 273; DOI: 10.1021/jm00314a039 |
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Salts of α-Amino-p-toluenesulfonamide Roman Rakoczy and Frederick C. Nachod pp 273 - 274; DOI: 10.1021/jm00314a040 |
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Bisoxime Sulfonates and Bisquaternary Hydrazones William A. Remers, Gabriel J. Gibs, and Martin J. Weiss pp 274 - 276; DOI: 10.1021/jm00314a041 |
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The Synthesis and Tranquilizer Activity of 2- and 4-Substituted 3,5-Morpholinediones Frank A. Baron, Calvin A. Vanderwerf, and David H. Tedeschi pp 276 - 279; DOI: 10.1021/jm00314a042 |
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Some Derivatives of 8-Thia-3-azabicyclo[3.2.1]octane F. Fried, Raj Nandan Prasad, and Alan P. Gaunce pp 279 - 281; DOI: 10.1021/jm00314a043 |
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Structure of Antibiotic C-73X Adorjan Aszalos, Herman Hoberecht, and Allen I. Cohen pp 281 - 284; DOI: 10.1021/jm00314a044 |
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5-Substituted Pyrimidines. II. The Synthesis of 2-Amino-4-hydroxy-6-methyl-5-(2-hydroxy-3-amino)propylpyrimidines A. M. Triggle and D. J. Triggle pp 285 - 285; DOI: 10.1021/jm00314a045 |
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Synthesis of N-(2-Chloroethyl)amides of Amino Acids as Potential Cytotoxic Agents Jiban K. Chakrabarti and Orrie M. Friedman pp 285 - 287; DOI: 10.1021/jm00314a046 |
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Synthesis of New Alkylating Agents Lise Nicole and Louis Berlinguet pp 287 - 288; DOI: 10.1021/jm00314a047 |
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1,3-Dimethyl-5-fluoro-6-azauracil and Some 5-Bromo-6-azauracil Derivatives G. J. Durr pp 288 - 289; DOI: 10.1021/jm00314a048 |
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cis-1-(3-Dimethylaminopropyl)-2,3- pentamethylenetetrahydroquinoline Walter F. Gannon pp 289 - 289; DOI: 10.1021/jm00314a049 |
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Preparation of Substituted Diaminopropanols F. C. Pennington, K. Mortenson, and B. W. Macharia pp 289 - 290; DOI: 10.1021/jm00314a050 |
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Orotic Acid Analogs. 2,5-Disubstituted 6-Hydroxy-4-carboxypyrimidines Saul Borodkin, Sigurdur Jonsson, George H. Cocolas, and Robert L. McKee pp 290 - 292; DOI: 10.1021/jm00314a051 |
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Routes to Unsymmetrical N,N′-Diarylethylenediamines C. H. Yoder and J. J. Zuckerman pp 292 - 292; DOI: 10.1021/jm00314a052 |
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Syntheses of Some Aminonaphythylalanines Joseph D. Benigni and R. L. Minnis pp 293 - 294; DOI: 10.1021/jm00314a053 |
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Some N-Substituted Derivatives of Bis(4-amino-3-nitrophenyl) Sulfone William F. Hart, Martin E. McGreal, Rita T. Enright, and Robert V. Mark pp 294 - 294; DOI: 10.1021/jm00314a054 |
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Research on Steroids. Volume II. Romano Deghenghi pp 295 - 295; DOI: 10.1021/jm00314a055 |
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Hypotensive Peptides. Philip A. Khairallah pp 295 - 295; DOI: 10.1021/jm00314a056 |
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Chemistry and Applied Pharmacology of Tranquilizers. A Primer for Students and Practitioners. Alfred Burger pp 295 - 295; DOI: 10.1021/jm00314a057 |
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Textbook of Biochemistry. Alfred Burger pp 296 - 296; DOI: 10.1021/jm00314a058 |
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Mikrobiologiczeskie Transformacii Steroidov (Microbiologica Transformations of Steroids). Eliahu Caspi pp 296 - 296; DOI: 10.1021/jm00314a059 |
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Irreversible Enzyme Inhibitors. LXXV.1,2 Inhibitors of Thymidine Phosphorylase. I. Mode of Ribofuranose Binding B. R. Baker pp 297 - 301; DOI: 10.1021/jm00315a001 |
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Irreversible Enzyme Inhibitors. LXXVI.1,2 Inhibitors of Thymidine Phosphorylase. II.2 Hydrophobic Bonding by 1-Substituted Uracils B. R. Baker and Mitsutaka Kawazu pp 302 - 304; DOI: 10.1021/jm00315a002 |
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Irreversible Enzyme Inhibitors. LXXVII.1,2 Inhibitors of Thymidine Phosphorylase. III.2 Hydrophobic Bonding by 1-Substituted Uracils Containing Additional Substituents at the 5 and 6 Positions B. R. Baker, Mitsutaka Kawazu, Daniel V. Santi, and Thomas J. Schwan pp 304 - 311; DOI: 10.1021/jm00315a003 |
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Irreversible Enzyme Inhibitors. LXXVIII.1,2 Inhibitors of Thymidine Phosphorylase. IV.2 Hydrophobic Bonding by Uracils Substituted at the 5 and 6 Positions B. R. Baker and Mitsutaka Kawazu pp 311 - 313; DOI: 10.1021/jm00315a004 |
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Irreversible Enzyme Inhibitors. LXXIX.1,2 Inhibitors of Thymidine Phosphorylase. V.2 Mode of Pyrimidine Binding B. R. Baker and Mitsutaka Kawazu pp 313 - 315; DOI: 10.1021/jm00315a005 |
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Irreversible Enzyme Inhibitors. LXXX.1,2 Inhibitors of Thymidine Phosphorylase. VI.2 Hydrophobic Bonding with 6 Substituents on the Acidic 5-Nitro- and 5-Bromouracils B. R. Baker and Mitsutaka Kawazu pp 316 - 320; DOI: 10.1021/jm00315a006 |
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Approaches to the Synthesis of 1-Deazauridine and 2′-Deoxy-1-deazauridine Mathias P. Mertes, James Zielinski, and Conrad Pillar pp 320 - 325; DOI: 10.1021/jm00315a007 |
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Pyrrolopyrimidine Nucleosides. I. The Synthesis of 4-Substituted 7-(β-D-Ribofuranosyl)pyrrolo[2,3-d]pyrimidines from Tubercidin John F. Gerster, Barbara Carpenter, Roland K. Robins, and Leroy B. Townsend pp 326 - 331; DOI: 10.1021/jm00315a008 |
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Nucleosides. V. 2-Thiopyrimidine β-D-Arabinofuranosides W. V. Ruyle and T. Y. Shen pp 331 - 334; DOI: 10.1021/jm00315a009 |
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Substituted 2,3-Dihydro-4(1H)-quinazolinones. A New Class of Inhibitors of Cell Multiplication Harry L. Yale and Marion Kalkstein pp 334 - 336; DOI: 10.1021/jm00315a010 |
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Tumor Inhibitors. XXIII.1 The Cytotoxic Principles of Marah oreganus H.2 S. Morris Kupchan, Allison H. Gray, and Michael D. Grove pp 337 - 340; DOI: 10.1021/jm00315a011 |
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Vitamin B2 Analogs. Synthesis and Biological Activity of Homologs of Pyridoxal 5′-Phosphate Peter F. Mühlradt, Y. Morino, and Esmond E. Snell pp 341 - 344; DOI: 10.1021/jm00315a012 |
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Synthesis and Antagonist Properties of Pyridoxol Analogs Modified in the 5 Position W. Korytnyk, B. Paul, A. Bloch, and C. A. Nichol pp 345 - 352; DOI: 10.1021/jm00315a013 |
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Diastereomers of 2-Amino-3-methylaminobutyric Acid, Aza Analogs of Isoleucine Tommy J. McCord, David C. Foyt, Joel L. Kirkpatrick, and Alvie L. Davis pp 353 - 355; DOI: 10.1021/jm00315a014 |
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Lincomycin. VI. 4′-Alkyl Analogs of Lincomycin. Relationship between Structure and Antibacterial Activity Barney J. Magerlein, Robert D. Birkenmeyer, and Fred Kagan pp 355 - 359; DOI: 10.1021/jm00315a015 |
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The 6-Deoxytetracyclines. IX. Imidomethylation Michael J. Martell, Adma S. Ross, and James H. Boothe pp 359 - 363; DOI: 10.1021/jm00315a016 |
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Semisynthetic Penicillins. IV. Pyridylmethylpenicillins and Related Cephalosporins R. John Stedman, Alice C. Swift, Libby S. Miller, Margaret M. Dolan, and John R. E. Hoover pp 363 - 366; DOI: 10.1021/jm00315a017 |
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5-Phenyl-2,4-pentadienamides as Potential Antimalarial Agents Leslie M. Werbel, Nancy Headen, and Edward F. Elslager pp 366 - 370; DOI: 10.1021/jm00315a018 |
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Metabolic Studies with Deuterated Phenobarbital James M. Perel, Peter G. Dayton, Carol L. Tauriello, Leonard Brand, and Lester C. Mark pp 371 - 374; DOI: 10.1021/jm00315a019 |
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Mass Spectrometric Identification of the Metabolites of Methyl N-(o-Aminophenyl)-N-(3-dimethylaminopropyl)anthranilate David L. Smith and Marvin F. Grostic pp 375 - 379; DOI: 10.1021/jm00315a020 |
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Some Derivatives of Metamorphinan Marshall Gates and David Arthur Klein pp 380 - 382; DOI: 10.1021/jm00315a021 |
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Benzomorphans. Optically Active and trans Isomers B. F. Tullar, L. S. Harris, R. L. Perry, Anne K. Pierson, A. E. Soria, W. F. Wetterau, and N. F. Albertson pp 383 - 386; DOI: 10.1021/jm00315a022 |
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Tremor-Producing Aminopropanols J. Kenneth Horner, Leon Otis, and W. A. Skinner pp 387 - 391; DOI: 10.1021/jm00315a023 |
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Aryloxyalkylaminoguanidines. Their Synthesis and Biological Properties J. Augstein, S. M. Green, A. M. Monro, T. I. Wrigley, A. R. Katritzky, and G. J. T. Tiddy pp 391 - 400; DOI: 10.1021/jm00315a024 |
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New Antihypertensive Aminoalkyltetrazoles Shin Hayao, Herbert J. Havera, Wallace G. Strycker, T. J. Leipzig, and Rodolfo Rodriguez pp 400 - 402; DOI: 10.1021/jm00315a025 |
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Synthesis and Pharmacology of Some Hydroxylated Tryptamines Robert G. Taborsky, Peter Delvigs, Djuro Palaic, and Merlin Bumpus pp 403 - 407; DOI: 10.1021/jm00315a026 |
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3-Aminoalkyl-2-benzoxazolinones Joseph Sam, C. W. Richmond, and J. L. Valentine pp 408 - 410; DOI: 10.1021/jm00315a027 |
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Isoxazoles. XVIII. Synthesis and Pharmacological Properties of 5-Aminoalkyl- and 3-Aminoalkylisoxazoles and Related Derivatives Hideo Kan[UNK]o, Ikuo Adachi, Ryonosuke Kido, and Katumi Hirose pp 411 - 418; DOI: 10.1021/jm00315a028 |
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Phenylindenes and Phenylindans with Antireserpine Activity Stanley J. Dykstra, James M. Berdahl, Kenneth N. Campbell, Charles M. Combs, and Donald G. Lankin pp 418 - 428; DOI: 10.1021/jm00315a029 |
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Substituted Anilinopyridine Carboxylic Acids with Antiinflammatory Activity D. Evans, K. S. Hallwood, C. H. Cashin, and H. Jackson pp 428 - 431; DOI: 10.1021/jm00315a030 |
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2,4,7-Triamino-6-ortho-substituted Arylpteridines. A New Series of Potent Antimalarial Agents T. S. Osdene, Peter B. Russell, and Leo Rane pp 431 - 434; DOI: 10.1021/jm00315a031 |
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Cyclopropylogs of Thyronine Derivatives Robert A. Pages and Alfred Burger pp 435 - 440; DOI: 10.1021/jm00315a032 |
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The Synthesis and Biological Evaluation of 16β-Amino-17α,20-dihydroxypregnanes Clarence G. Bergstrom pp 440 - 445; DOI: 10.1021/jm00315a033 |
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Totally Synthetic Hormones. XVI.1 The Conversion of Estr-4-en-17β-ol to Testosterone and the Total Synthesis of Some 18-Methylandrostane and 18-Methylpregnane Derivatives D. P. Strike, D. Herbst, and Herchel Smith pp 446 - 451; DOI: 10.1021/jm00315a034 |
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8-Aza Steroids. IV.1 8-Aza-19-norprogestogens Richard E. Brown, David M. Lustgarten, R. John Stanaback, and Robert I. Meltzer pp 451 - 456; DOI: 10.1021/jm00315a035 |
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Insect Chemosterilants. V. Derivatives of Melamine Alexej B. Bořkovec and Albert B. DeMilo pp 457 - 461; DOI: 10.1021/jm00315a036 |
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Sulfonanilides. II. Analogs of Catecholamines A. A. Larsen, William A. Gould, Herbert R. Roth, William T. Comer, Robert H. Uloth, K. W. Dungan, and P. M. Lish pp 462 - 472; DOI: 10.1021/jm00315a037 |
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Studies on Latent Derivatives of Aminoethanethiols as Potentially Selective Cytoprotectants. VI. Synthesis of N-(2-Mercaptoethyl)carbamoylamino Acids Ezra Khedouri, Vytautas Grubliauskas, and Orrie M. Friedman pp 472 - 474; DOI: 10.1021/jm00315a038 |
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Some Biologically Active N6-Methylated Adenosine Analogs G. Gough and M. Helen Maguire pp 475 - 478; DOI: 10.1021/jm00315a039 |
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Unnatural Amino Acids. II. Congeners of DL-3-Carboxy-4-methoxyphenylalanine Frederick Leonard, Abraham Wajngurt, Walter Tschannen, and M. Klein pp 478 - 481; DOI: 10.1021/jm00315a040 |
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Synthesis of Potential Antineoplastic Agents. XVII. N,N-Bis(2-fluoroethyl)anilines Frank D. Popp, Fredrick P. Silver, and Dru W. Alwani pp 481 - 484; DOI: 10.1021/jm00315a041 |
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4-Hydroxy-2-butanone Thiosemicarbazone, a Potential Anticancer Agent Benjamin Prescott pp 484 - 485; DOI: 10.1021/jm00315a042 |
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The 6-Deoxytetracyclines. VIII. Acylaminomethylamides Michael J. Martell, Adma S. Ross, and James H. Boothe pp 485 - 486; DOI: 10.1021/jm00315a043 |
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1,3,2-Diazaphosphorine 2-Oxides. IV.1 A New Method for the Preparation of 2-(N-Arylamino)-and 2-(N-Alkylamino)-1,3,2-diazaphosphorine 2-Oxides2 John H. Billman and Ralph F. May pp 486 - 488; DOI: 10.1021/jm00315a044 |
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Scopoletin, an Antispasmodic Component of Viburnum opulus and prunifolium Charles H. Jarboe, Karimullah A. Zirvi, John A. Nicholson, and Charlotte M. Schmidt pp 488 - 489; DOI: 10.1021/jm00315a045 |
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Synthesis of Substituted 2-(2-Biphenylyl)ethylamines as Potential Analgeties George Tsatsas, Avra Parrea-Sandris, and Constantine Sandris pp 489 - 491; DOI: 10.1021/jm00315a046 |
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Analogs of 2,6-Pyridinedimethanol Bis(N-methylcarbamate) P. F. Juby, R. B. Babel, G. E. Bocian, N. M. Cladel, J. C. Godfrey, B. A. Hall, T. W. Hudyma, G. M. Luke, J. D. Matiskella, W. F. Minor, T. A. Montzka, R. A. Partyka, R. T. Standridge, and L. C. Cheney pp 491 - 495; DOI: 10.1021/jm00315a047 |
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2-Acylimino-1,1-dimethylphenethylamines and Related Compounds. Anoreetic Agents John Krapcho and John P. High pp 495 - 497; DOI: 10.1021/jm00315a048 |
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5-(3-Dimethylaminopropyl)-2,8-diaza-10, 11-dihydro-5H-dibenzo[b,f]azepine Frank J. Villani pp 497 - 498; DOI: 10.1021/jm00315a049 |
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2-Phenylindolizines Lewis. A. Walter and Phyllis Margolis pp 498 - 499; DOI: 10.1021/jm00315a050 |
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N-(ω-Aminoalkoxy)phthalimides Milton J. Kornet and Anthony Wu pp 499 - 500; DOI: 10.1021/jm00315a051 |
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The Synthesis of Aryloxybiguanide and Aryloxyguanidine Salts William J. Fanshawe and Victor J. Bauer pp 500 - 501; DOI: 10.1021/jm00315a052 |
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Reactions of Phenacyl Sulfides with Ammonia, Amines, and Hydrazines Carl R. Johnson and Ishai Sataty pp 501 - 503; DOI: 10.1021/jm00315a053 |
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Steroidal 2,3-Epithiospirolactones P. D. Klimstra pp 503 - 505; DOI: 10.1021/jm00315a054 |
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3,4-Dihydro-1,3-oxazines from Dcycloheexylcarbodiimide Everette L. May pp 505 - 506; DOI: 10.1021/jm00315a055 |
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Terpene Compounds as Drugs. II. Terpenyl Derivatives of Barbituric Acids and Normeperidine Gianfranco Pala, Elda Crescenzi, and Tiberio Bruzzese pp 507 - 508; DOI: 10.1021/jm00315a056 |
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Terpenes as Drugs. I. 1-Terpenyl-3-arylsulfonylureas Gianfranco Pala, Antonio Mantegani, and Germano Coppi pp 508 - 508; DOI: 10.1021/jm00315a057 |
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Potential Antimalarial Substances. Amides of o-Ethoxy- and p-Isopropylbenzoic Acids Leslie M. Werbel, Carolyn A. Hess, and Edward F. Elslager pp 508 - 509; DOI: 10.1021/jm00315a058 |
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4-(1-Methyl-4-pyrrolidinobutylamino)-7-chloroquinoline and 4-(1-Methyl-4-morpholinobutylamino)-7-chloroquinoline as Potential Antimalarials Peter K. Iber and Betty J. Boone pp 509 - 510; DOI: 10.1021/jm00315a059 |
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Substituted N-Aminomethylisatins Rajendra S. Varma and W. Lewis Nobles pp 510 - 510; DOI: 10.1021/jm00315a060 |
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Synthesis of Potential Anticancer Agents Charles E. Williamson, Thomas J. Sayers, Arnold M. Seligman, and Benjamin Witten pp 511 - 511; DOI: 10.1021/jm00315a061 |
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The Synthesis of Aryloxycarbamates Victor J. Bauer, Harry P. Dalalian, and William J. Fanshawe pp 512 - 512; DOI: 10.1021/jm00315a062 |
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The Salicylates. A Critical Bibliographical Review. Alfred Burger pp 512 - 512; DOI: 10.1021/jm00315a063 |
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Naphthoquinone Antimalarials. XXIX. 2-Hydroxy-3-(ω-cyclohexylalkyl)-1,4-naphthoquinones Louis F. Fieser, Joseph P. Schirmer, Sydney Archer, Roman R. Lorenz, and Peter I. Pfaffenbach pp 513 - 517; DOI: 10.1021/jm00316a001 |
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Naphthoquinone Antimalarials. XXX.1 2-Hydroxy-3-[ω-(1-adamantyl)alkyl]-1,4-naphthoquinones2 Louis F. Fieser and Musa Z. Nazer pp 517 - 521; DOI: 10.1021/jm00316a002 |
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Potential Antimalarial Compounds.1 IX.2 Pyrimidine Derivatives of Urea and Guanidine Tadeusz Urbański, Barbara Serafin, and Jerzy Żylowski pp 521 - 525; DOI: 10.1021/jm00316a003 |
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An Apparent Correlation between the in Vitro Activity of Chloramphenicol Analogs and Electronic Polarizability Arthur Cammarata pp 525 - 527; DOI: 10.1021/jm00316a004 |
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Structure and Properties of Sulfones. I. Electric Moment of 4,4′-Diaminodiphenyl Sulfone Judith A. Singer, William P. Purcell, and Clifton C. Thompson pp 528 - 529; DOI: 10.1021/jm00316a005 |
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Antibacterial Nitrofuran Derivatives. I. 5-Nitro-2-furaldehyde Semicarbazones and Thiosemicarbazones D. Nardi, E. Massarani, A. Tajana, L. Degen, and M. J. Magistretti pp 530 - 533; DOI: 10.1021/jm00316a006 |
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Insect Sex Attractants. VI. 7-Dodecen-1-ol Acetates and Congeners Nathan Green, Martin Jacobson, Thomas J. Henneberry, and Albert N. Kishaba pp 533 - 535; DOI: 10.1021/jm00316a007 |
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Organic Fluorine Compounds. III. Action of Perchloryl Fluoride on Substituted Ethyl Cyanoacetates and Animal Toxicities of the Fluorinated Products1-3 Herman Gershon, Stephen G. Schulman, and A. David Spevack pp 536 - 541; DOI: 10.1021/jm00316a008 |
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Antiinflammatory Dialkylaminoalkylureas William E. Coyne and John W. Cusic pp 541 - 546; DOI: 10.1021/jm00316a009 |
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Some Steroidal Cyclic Ethers As Antiestrogens Edward A. Brown pp 546 - 551; DOI: 10.1021/jm00316a010 |
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6-Chloro-6-dehydro-A-nor Steroids with Progestational Activity. 7α-Chloro-A-nor Steroids Patrick A. Diassi, Seymour D. Levine, and Raymond M. Palmere pp 551 - 556; DOI: 10.1021/jm00316a011 |
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The Synthesis of Hydroxylamine Derivatives Possessing Hypocholesteremic Activity B. J. Ludwig, F. Dürsch, M. Auerbach, K. Tomeczek, and F. M. Berger pp 556 - 564; DOI: 10.1021/jm00316a012 |
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2-(2-Pyridyl)-1,2-diarylalkanols as Hypocholesteremic Agents J. H. Burckhalter, William D. Dixon, Martin L. Black, Roger D. Westland, Leslie M. Werbel, Horace A. DeWald, John R. Dice, Gertrude Rodney, and Donald H. Kaump pp 565 - 575; DOI: 10.1021/jm00316a013 |
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Imidazoline Derivatives with Antiarrhythmic Activity L. H. Werner, S. Ricca, A. Rossi, and George deStevens pp 575 - 582; DOI: 10.1021/jm00316a014 |
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Cassaine Analogs. II. 7-Deoxy Basic Esters Robert L. Clarke, Sol J. Daum, Philip E. Shaw, Theodore G. Brown, G. E. Groblewski, and W. V. O'Connor pp 582 - 593; DOI: 10.1021/jm00316a015 |
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Cassaine Analogs. IV. Distant Analogs of Cassaine Robert L. Clarke, Sol J. Daum, Philip E. Shaw, Theodore G. Brown, G. E. Groblewski, and W. V. O'Connor pp 593 - 597; DOI: 10.1021/jm00316a016 |
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Pyrazine Diuretics. III. 5- and 6-Alkyl, -Cycloalkyl, and -Aryl Derivatives of N-Amidino-3-aminopyrazinecarboxamides John B. Bicking, Charles M. Robb, Sara F. Kwong, and Edward J. Cragoe pp 598 - 602; DOI: 10.1021/jm00316a017 |
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The Adamantyl Group in Medicinal Agents. IV. Sedative Action of 3,5,7-Trimethyladamantane-1-carboxamide1 and Related Agents Koert Gerzon, Donald J. Tobias, Richard E. Holmes, Robert E. Rathbun, and Richard W. Kattau pp 603 - 606; DOI: 10.1021/jm00316a018 |
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The Anticonvulsant Activity of 4a,8a-Naphthalenedicarboximide and Its Derivatives Eugene R. Wagner and Allan D. Rudzik pp 607 - 611; DOI: 10.1021/jm00316a019 |
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Preparation and Anticonvulsant Activity of Some Aryldialkylsuccinimides Fred P. Hauck, JoAnn Demick, and Jane Fan pp 611 - 614; DOI: 10.1021/jm00316a020 |
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Pharmacologically Active Acetylene Compounds. I.1,2 Structural Modifications of Oxotremorine John L. Neumeyer, Urve V. Moyer, Janice A. Richman, Frank J. Rosenberg, and David G. Teiger pp 615 - 620; DOI: 10.1021/jm00316a021 |
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ω-Azabicyclic Butyrophenones Charles H. Grogan and Leonard M. Rice pp 621 - 623; DOI: 10.1021/jm00316a022 |
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Structure and Biological Activity of Some Reduction Products of Strychnine, Brucine, and Their Congeners Richard Rees and Herchel Smith pp 624 - 627; DOI: 10.1021/jm00316a023 |
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New Psychotropic Agents. VIII.1 Analogs of Amitriptyline Containing the Normeperidine Group M. A. Davis, F. Herr, R. A. Thomas, and Marie-Paule Charest pp 627 - 635; DOI: 10.1021/jm00316a024 |
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Neuropharmacological Investigation of N-Benzylsulfamides Paul Aeberli, John Gogerty, and William J. Houlihan pp 636 - 642; DOI: 10.1021/jm00316a025 |
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Synthesis of Some Dibenzo[b,f][1,5]diazocines and Dibenzo[b,f][1,4]diazocines John G. Topliss, Elizabeth P. Shapiro, and Robert I. Taber pp 642 - 646; DOI: 10.1021/jm00316a026 |
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Synthesis and Biological Activity of Some Ring-Substituted Tryptamines R. R. Hunt and R. W. Brimblecombe pp 646 - 648; DOI: 10.1021/jm00316a027 |
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The 2-Thiopseudourea [ILL], a New Local Anesthesiophore B. M. Regan, F. T. Galysh, and R. N. Morris pp 649 - 652; DOI: 10.1021/jm00316a028 |
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Thyromimetics. VII. Isopropyl Analogs of Thyroid Hormones Benjamin Blank and Francis R. Pfeiffer pp 653 - 656; DOI: 10.1021/jm00316a029 |
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Structure-Activity Relations in the Vitamin E Series.1 I. Effects of 5-Methyl Substitution on 6-Hydroxy-2,2,5,7,8-pentamethylchroman W. A. Skinner, R. M. Parkhurst, J. Scholler, P. Alaupovic, Q.E. Crider, and K. Schwarz pp 657 - 661; DOI: 10.1021/jm00316a030 |
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Synthesis of 3-Indolyl and 5-Bromo-3-indolyl Phosphate for Histochemical Demonstration of Alkaline Phosphatase K. C. Tsou, Helen C. F. Su, Dorothy J. Rabiger, Hans Heymann, and Arnold M. Seligman pp 662 - 664; DOI: 10.1021/jm00316a031 |
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Analogs of Tubercidin John A. Montgomery and Kathleen Hewson pp 665 - 667; DOI: 10.1021/jm00316a032 |
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The Modes of Decomposition of 1,3-Bis(2-chloroethyl)-1-nitrosourea and Related Compounds John A. Montgomery, Ruby James, George S. McCaleb, and Thomas P. Johnston pp 668 - 674; DOI: 10.1021/jm00316a033 |
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The Synthesis of Potential Anticancer Agents. XXXVII. N-Nitrosoureas. III. 1,5-Bis(2-chloroethyl)-1-nitrosobiuret and Related Derivatives of Biurets, Biureas, and Carboxamides Thomas P. Johnston and Pamela S. Opliger pp 675 - 681; DOI: 10.1021/jm00316a034 |
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Irreversible Enzyme Inhibitors. XCV. 8-(m-Bromoacetamidobenzylthio)hypoxanthine, an Active-Site-Directed Irreversible Inhibitor of Xanthine Oxidase1-3 B. R. Baker and Janos Kozma pp 682 - 685; DOI: 10.1021/jm00316a035 |
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Enzyme Inhibitors. XVII. Kinetic Studies on the Irreversible Inhibition of Adenosine Deaminase Howard J. Schaeffer, Michael A. Schwartz, and Eugene Odin pp 686 - 689; DOI: 10.1021/jm00316a036 |
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Enzyme Inhibitors. XVIII. Studies on the Stereoselectivity of Inhibition of Adenosine Deaminase by DL-, D-, and L-9-(2-Hydroxypropyl)adenine Howard J. Schaeffer and Robert Vince pp 689 - 691; DOI: 10.1021/jm00316a037 |
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Antineoplastic Agents. XVIII. N-(2-Haloethyl)benzylamines G. R. Pettit, S. K. Gupta, and P. A. Whitehouse pp 692 - 696; DOI: 10.1021/jm00316a038 |
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Alkylating Agents Related to 2,2′-Biaziridine. I. Compounds Derived from 1,4-Diamino-2,3-butanediol Peter W. Feit and Ole Tvaermose Nielsen pp 697 - 700; DOI: 10.1021/jm00316a039 |
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Potential Carcinolytic Agents.1,2 V. Enamine Mustards Zinon B. Papanastassiou, Robert J. Bruni, and Edward V. White V pp 701 - 706; DOI: 10.1021/jm00316a040 |
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Potential Antitumor Agents. V. Bisquaternary Salts G. J. Atwell and B. F. Cain pp 706 - 713; DOI: 10.1021/jm00316a041 |
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Penetration of Brain and Brain Tumor. VII. Tumor-Binding Sulfhydryl Boron Compounds A. H. Soloway, H. Hatanaka, and M. A. Davis pp 714 - 717; DOI: 10.1021/jm00316a042 |
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Maleamic Acids That Affect Plasma Cholesterol and Penicillin Excretion Everett M. Schultz, William A. Bolhofer, Albert Augenblick, John B. Bicking, Charles N. Habecker, J. Kenneth Horner, Sara F. Kwong, and Adolph M. Pietruszkiewicz pp 717 - 724; DOI: 10.1021/jm00316a043 |
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The Stereochemistry of 2,3-Diphenyl-1-methylpropylamine Seemon H. Pines, John M. Chemerda, Matthew A. Kozlowski, Leonard M. Weinstock, Paul Davis, Barry Handelsman, Victor J. Grenda, and Glenn W. Lindberg pp 725 - 728; DOI: 10.1021/jm00316a044 |
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The Syntheses of 4′-Bromo-10-methyl-1,2-benzanthracene and 4′-Chloro-10-methyl-1,2-benzanthracene Melvin S. Newman and N. Venkateswaran pp 728 - 729; DOI: 10.1021/jm00316a045 |
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Metabolism of 2-Diethylamino-6,7-dimethoxy-4(3H)-quinazolinone M. Schach von Wittenau and Timothy F. Brewer pp 729 - 730; DOI: 10.1021/jm00316a046 |
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Carboranes. III. Boron-Containing Acridines M. A. Davis and A. H. Soloway pp 730 - 732; DOI: 10.1021/jm00316a047 |
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N-(4-Biphenyl)-N-(2-diethylaminoethyl)-mandelamide Hydrochloride. A Potent Local Anesthetic for Use with Sulfhydryl Inhibitors for Cancer Therapy Frances E. Knock pp 733 - 733; DOI: 10.1021/jm00316a048 |
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Sulfate Esters of 5-Iododeoxyuridine and 5-Iododeoxycytidine Pauline K. Chang, Louis J. Sciarini, and John W. Cramer pp 733 - 735; DOI: 10.1021/jm00316a049 |
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Potential Carcinostatic Agents. I. Derivatives and Analogs of 1-(2-Hydroxyethyl)-3-(4-tolyl)urea Harold G. Nelson, Frederic J. Shelton, and William H. Wetzel pp 735 - 736; DOI: 10.1021/jm00316a050 |
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The Preparation of Some Antimalarials with Quaternary Carbon Side Chains D. E. Pearson and J. C. Craig pp 737 - 737; DOI: 10.1021/jm00316a051 |
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Nitrofuryl Heterocycles. VI.1 l-Alkyl-and l-Aryl-5-(5-nitro-2-furyl)tetrazoles Harry R. Snyder pp 737 - 739; DOI: 10.1021/jm00316a052 |
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2-(Purin-6-yl)-2-thiopseudourea Hydrochloride Eugene F. McInerney and Eugene J. Kupchik pp 739 - 740; DOI: 10.1021/jm00316a053 |
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2-(Purin-6-yl)-2-thiopseudourea Hydrochloride Eugene F. McInerney and Eugene J. Kupchik pp 741 - 741; DOI: 10.1021/jm00316a054 |
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Eugenolglycolic Acid Derivatives Noël J. de Souza, A. N. Kothare, and V. V. Nadkarny pp 741 - 743; DOI: 10.1021/jm00316a055 |
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A Ready Synthesis of Pantothenoylcystine J. F. Cavalla pp 743 - 743; DOI: 10.1021/jm00316a056 |
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Annual Reports in Medicinal Chemistry, 1965. Alfred Burger pp 744 - 744; DOI: 10.1021/jm00316a057 |
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Mechanisms of Release of Biogenic Amines. Alfred Burger pp 744 - 744; DOI: 10.1021/jm00316a058 |
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Progress in Drug Research. Volume 9. Henry G. Mautner pp 744 - 744; DOI: 10.1021/jm00316a059 |
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Lipoide. Alfred Burger pp 744 - 744; DOI: 10.1021/jm00316a060 |
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The Structure-Activity Relationship in Barbiturates and Its Similarity to That in Other Narcotics Corwin Hansch and Susan M. Anderson pp 745 - 753; DOI: 10.1021/jm00317a001 |
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Hückel Molecular Orbital Calculations for Some Antimalarial Drugs and Related Molecules Judith A. Singer and William P. Purcell pp 754 - 762; DOI: 10.1021/jm00317a002 |
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Nucleic Acids. I. The Synthesis of Nucleotides and Dinucleoside Phosphates Containing ara-Cytidine William J. Wechter pp 762 - 773; DOI: 10.1021/jm00317a003 |
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Nucleic Acids. II. Cytotoxicity Studies with Nucleotides and Dinucleoside Phosphates Containing ara-Cytidine Charles G. Smith, Harold H. Buskirk, and William L. Lummis pp 774 - 776; DOI: 10.1021/jm00317a004 |
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Nucleic Acids. III. Antiviral Activity of Nucleotides and Dinucleoside Phosphates Containing ara-Cytidine H. E. Renis, C. A. Hollowell, and G. E. Underwood pp 777 - 782; DOI: 10.1021/jm00317a005 |
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Totally Synthetic Steroid Hormones. XVII.1 Further Studies on the Synthesis of dl-18-Methylandrostane and dl-18-Methylpregnane Derivatives Richard Rees, D. P. Strike, and Herchel Smith pp 783 - 789; DOI: 10.1021/jm00317a006 |
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The Synthesis of Certain 17α-Alkyl Corticoids Robert E. Schaub and Martin J. Weiss pp 789 - 795; DOI: 10.1021/jm00317a007 |
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Some 17α-Cyclopropyl Steroids John W. Dean, Gordon O. Potts, and Robert G. Christiansen pp 795 - 799; DOI: 10.1021/jm00317a008 |
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Steroids Possessing Nitrogen Atoms. III. Synthesis of New Highly Active Corticoids. [17α,16α,-d]Oxazolino Steroids Giangiacomo Nathansohn, Giorgio Winters, and Emilio Testa pp 799 - 802; DOI: 10.1021/jm00317a009 |
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Nonsteroidal Hypocholesteremic Agents. I. The Synthesis and Serum Sterol Lowering Properties of Substituted 4-(2-Dialkylaminoethoxy)diphenylamines and Related Compounds Frederick L. Bach, John C. Barclay, and Elliott Cohen pp 802 - 806; DOI: 10.1021/jm00317a010 |
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1-[5-Arylfurfurylidene)amino]hydantoins. A New Class of Muscle Relaxants Harry R. Snyder, Charles S. Davis, Robert K. Bickerton, and Robert P. Halliday pp 807 - 810; DOI: 10.1021/jm00317a011 |
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The Metabolic Fate of Some Silicon-Containing Carbamates Ralph J. Fessenden and Charles Ahlfors pp 810 - 812; DOI: 10.1021/jm00317a012 |
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Compounds Acting on the Central Nervous System. VII. Studies in 1-Pyridyl-4-substituted Piperazines. A New Class of Anticonvulsants P. C. Jain, V. Kapoor, Nitya Anand, A. Ahmad, and G. K. Patnaik pp 812 - 818; DOI: 10.1021/jm00317a013 |
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1-Amino-4-aryl-4-piperidinols as Potential Antidepressants N. J. Harper, C. W. T. Hussey, M. E. Peel, A. C. Ritchie, and Juliet M. Waring pp 819 - 822; DOI: 10.1021/jm00317a014 |
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1-(3-Dimethylaminopropyl)-2-methyl-2-phenyl-1-indanol and Related Compounds. A New Class of Analgesic Agents Chester F. Turk and John Krapcho pp 823 - 825; DOI: 10.1021/jm00317a015 |
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Compounds Affecting the Central Nervous System. IV. Substituted 2-Benzyl-3-dialkylaminoalkylindenes and Related Compounds C. R. Ganellin, J. M. Loynes, H. F. Ridley, and R. G. W. Spickett pp 826 - 833; DOI: 10.1021/jm00317a016 |
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Sympathetic Nervous System Blocking Agents. III. Derivatives of Benzylguanidine1-3 James H. Short and Thomas D. Darby pp 833 - 840; DOI: 10.1021/jm00317a017 |
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Hypotensive 1,2-Benzisothiazole 1,1-Dioxides. I. Pyrazole and Pyrazoline Derivatives John J. Traverso, Calvert W. Whitehead, James F. Bell, Harold E. Boaz, and Paul W. Willard pp 840 - 844; DOI: 10.1021/jm00317a018 |
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Hypotensive 1,2-Benzisothiazole 1,1-Dioxides. II. 3-Hydrazino-1,2-benzisothiazole 1,1-Dioxides and their Hydrazone and Amide Derivatives Calvert W. Whitehead, John J. Traverso, James F. Bell, and Paul W. Willard pp 844 - 849; DOI: 10.1021/jm00317a019 |
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Hypotensive 1,2-Benzisothiazole 1,1-Dioxides. III. 3-[2-(2-Methyl-2-butylidene)hydrazino]-1,2-benzisothiazole 1,1-Dioxide and Related Analogs Paul W. Willard, Calvert W. Whitehead, and John J. Traverso pp 849 - 852; DOI: 10.1021/jm00317a020 |
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A New Class of Potent Decarboxylase Inhibitors. β-(3-Indolyl)-α-hydrazinopropionic Acids Edward J. Glamkowski, George Gal, Meyer Sletzinger, Curt C. Porter, and L. Sherman Watson pp 852 - 855; DOI: 10.1021/jm00317a021 |
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Synthesis of Some 3-Indenealkylamines. Comparison of the Biological Activity of 3-Indenealkylamines and 3-Benzo[b]thiophenealkylamines with Their Tryptamine Isosteres J. C. Winter, P. K. Gessner, and D. D. Godse pp 856 - 859; DOI: 10.1021/jm00317a022 |
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Metabolic Fate of Methoxamine and N-Isopropylmethoxamine A. Klutch and M. Bordun pp 860 - 863; DOI: 10.1021/jm00317a023 |
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Local Anesthetics with Enhanced Affinity for Proteins J. Hollowood, A. B. A. Jansen, and P. J. Southgate pp 863 - 867; DOI: 10.1021/jm00317a024 |
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Hycanthone,1 a New Active Metabolite of Lucanthone2 D. Rosi, G. Peruzzotti, E. W. Dennis, D. A. Berberian, H. Freele, B. F. Tullar, and S. Archer pp 867 - 876; DOI: 10.1021/jm00317a025 |
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Preparation and Schistosomicidal Activity of Some 4-Hydroxymethyl-3-chloroanilines D. Rosi, T. R. Lewis, R. Lorenz, H. Freele, D. A. Berberian, and S. Archer pp 877 - 880; DOI: 10.1021/jm00317a026 |
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Adrenergic Neurone Blocking Agents. II.1 Some Dioxane-Substituted Derivatives of Guanoxan A. M. Monro, G. W. H. Potter, and M. J. Sewell pp 880 - 883; DOI: 10.1021/jm00317a027 |
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as-Triazines. I. 5-Sulfanilamido Derivatives and Intermediates W. E. Taft and R. G. Shepherd pp 883 - 887; DOI: 10.1021/jm00317a028 |
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Synthesis of p-Acyl Analogs of Chloramphenicol and Their Antimicrobial Properties Maximilian von Strandtmann, George Bobowski, and John Shavel pp 888 - 890; DOI: 10.1021/jm00317a029 |
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Nitroimidazole Derivatives. Relationship between Structure and Antitrichomonal Activity K. Butler, H. L. Howes, J. E. Lynch, and D. K. Pirie pp 891 - 897; DOI: 10.1021/jm00317a030 |
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Anthelmintic Quaternary Salts. Thiacyanines and Hemithiacyanines D. L. Garmaise, C. H. Chambers, J. Komlossy, and R. C. McCrae pp 897 - 899; DOI: 10.1021/jm00317a031 |
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Pyrazine Diuretics. IV. N-Amidino-3-amino-6-substituted Pyrazinecarboxamides James H. Jones, John B. Bicking, and Edward J. Cragoe pp 899 - 903; DOI: 10.1021/jm00317a032 |
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Synthesis and Inhibitory Activity of Polyaspartic Acid Derivatives H. Nagy Kovacs, J. Kovacs, M. A. Pisano, and B. A. Shidlovsky pp 904 - 908; DOI: 10.1021/jm00317a033 |
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The Role of the 5′-Hydroxyl Group of Adenosine in Determining Substrate Specificity for Adenosine Deaminase Alexander Bloch, Morris J. Robins, and James R. McCarthy pp 908 - 912; DOI: 10.1021/jm00317a034 |
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Differential Binding to the Hydrophobic Bonding Region of T2 Phage Induced, Escherichia coli B, and Pigeon Liver Dihydrofolic Reductases B. R. Baker pp 912 - 917; DOI: 10.1021/jm00317a035 |
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Synthesis of Potential Anticancer Agents. XVIII. Nitrogen Mustards from 6-Substituted Coumarins Robert C. Elderfield and J. Roy pp 918 - 921; DOI: 10.1021/jm00317a036 |
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Synthesis of Potential Anticancer Agents. XIX. Nitrogen Mustards from 7-Hydroxycoumarin Derivatives Robert C. Elderfield and A. C. Mehta pp 921 - 923; DOI: 10.1021/jm00317a037 |
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Phosphorus-Nitrogen Compounds. VII.1,2 Urea, Aziridinecarboxamide, and Semicarbazide Derivatives Lindley A. Cates pp 924 - 927; DOI: 10.1021/jm00317a038 |
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Alkylating Agents Related to 2,2′-Biaziridine. II.1 N,N′-Dicarbethoxy-2,2′-biaziridine Peter W. Feit and Ole Tvaermose Nielsen pp 927 - 932; DOI: 10.1021/jm00317a039 |
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Syntheses of Metabolites of 7,12-Dimethylbenz[a]anthracene. 4-Hydroxy-7,12-dimethylbenz[a]anthracene, 7-Hydroxymethyl-12-methylbenz[a]anthracene, Their Methyl Ethers, and Acetoxy Derivatives James W. Flesher, Soekeni Soedigdo, and Donald R. Kelley pp 932 - 936; DOI: 10.1021/jm00317a040 |
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Derivatives of Fluorene. XXIII.1 New Thiofluorenes Related to Metabolism of the Carcinogen N-2-Fluorenylacetamide T. Lloyd Fletcher, Moses J. Namkung, and Hsi-Lung Pan pp 936 - 941; DOI: 10.1021/jm00317a041 |
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Substituted 2-Oxazolidinethiones Herman J. Eichel, Ronald J. Meyer, and Paul F. Buzzi pp 942 - 944; DOI: 10.1021/jm00317a042 |
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Agents Acting on the Central Nervous System. X. 1-Substituted 3-Phenyl-2,3,4,5-tetrahydro-1H-1-benzazepines J. M. Khanna and Nitya Anand pp 944 - 945; DOI: 10.1021/jm00317a043 |
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Amides and Esters of Benzo[b]thiophene-2-carboxylic Acid E. Campaigne and T. Bosin pp 945 - 946; DOI: 10.1021/jm00317a044 |
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Synthesis and Preliminary Pharmacological Evaluation of a Series of N,N′-Arylidenebis(acid amides) Theron A. Ebel, Arthur A. Harwood, and Allan M. Burkman pp 946 - 949; DOI: 10.1021/jm00317a045 |
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Effect of Organic Compounds on Reproductive Processes. VI. Alkylating Agents Derived from Various Diamines W. A. Skinner, J. Lange, T. E. Shellenberger, and W. T. Colwell pp 949 - 950; DOI: 10.1021/jm00317a046 |
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3-Halogenated Thyronines Paul Block pp 950 - 953; DOI: 10.1021/jm00317a047 |
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N,N′-Dimethyl-1-phenyl-1,2-propanediamine. A Hitherto Unreported Product in Ephedrine Synthesis Seymour Hyden, Santo Emmanuele, Henry Wetstein, and Godfrey Wilbert pp 953 - 954; DOI: 10.1021/jm00317a048 |
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4-Anilinopyrimidine-5-carboxylic Acids and Esters with Antiinflammatory and Analgetic Properties P. F. Juby and T. W. Hudyma pp 954 - 957; DOI: 10.1021/jm00317a049 |
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Derivatives of Fluorene. XXIV.1 Synthesis and Antitumor Activities of Some Imidazolidine-2,5-diones Hsi-Lung Pan and T. Lloyd Fletcher pp 957 - 959; DOI: 10.1021/jm00317a050 |
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Drug Latentiation. II.1 Labile Ether Derivatives of Phenolic Analgesics S. Morris Kupchan and Alan F. Casy pp 959 - 960; DOI: 10.1021/jm00317a051 |
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Drug Latentiation. III.1 Labile Amide Derivatives of Normeperidine S. Morris Kupchan and Allen C. Isenberg pp 960 - 961; DOI: 10.1021/jm00317a052 |
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DL-4,5-Dihydroxy-2-pyridylalanine, an Analog of 3,4-Dihydroxyphenylalanine S. J. Norton and Edward Sanders pp 961 - 963; DOI: 10.1021/jm00317a053 |
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Synthetic Biologically Active Polymers. IV. N1-Acylsulfanilamide-Formaldehyde Copolymers John R. Dombroski, L. Guy Donaruma, and John Razzano pp 963 - 964; DOI: 10.1021/jm00317a054 |
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Synthetic Biologically Active Polymers. V. 4,4′-Diaminodiphenyl Sulfone-Formaldehyde Copolymer John R. Dombroski, L. Guy Donaruma, and John Razzano pp 964 - 965; DOI: 10.1021/jm00317a055 |
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N-Thymidylglycine and Ethyl p-N-Thymidylaminobenzoate Mathias P. Mertes and Quentin Gilman pp 965 - 966; DOI: 10.1021/jm00317a056 |
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Chemistry of Cephalosporin Antibiotics. X.1 Synthesis of Methyl 3-Formyl-7-(thiophene-2-acetamido)-3-cephem-4-carboxylate, a New Cephalosporin Derivative J. W. Chamberlin and J. B. Campbell pp 966 - 968; DOI: 10.1021/jm00317a057 |
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Synthesis of α-Methyl-DLg-glutathione Daniel F. Veber, Karl Pfister, and Ralph Hirschmann pp 968 - 969; DOI: 10.1021/jm00317a058 |
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Synthesis of 5-Carboxy-2′-deoxyuridine Norbert Isenberg and Charles Heidelberger pp 970 - 971; DOI: 10.1021/jm00317a059 |
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Preparation and Properties of Clamoxyquin Pamoate,1 an Antiamebic and Antidiarrheal Agent Edward F. Elslager and Donald F. Worth pp 971 - 972; DOI: 10.1021/jm00317a060 |
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Synthesis and Antiviral and Antibacterial Activity of Certain N-Dialkylaminomethylisatin β-Thiosemicarbazones Rajendra S. Varma and W. Lewis Nobles pp 972 - 974; DOI: 10.1021/jm00317a061 |
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2,4-Bis(arylamino)-5-methylpyrimidines as Antimicrobial Agents Dolly Ghosh and Mina Mukherjee pp 974 - 975; DOI: 10.1021/jm00317a062 |
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Tumor Localizing Agents. II. Radioiodinated Analogs of 1,1-Dichloro-2,2-bis(chlorophenyl)ethane R. E. Counsell, R. E. Willette, and W. DiGuilio pp 975 - 977; DOI: 10.1021/jm00317a063 |
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Tumor Inhibitors. XXV. The Synthesis and Evaluation of 9-Nitro-1,2,3,4-tetrahydrophenanthrene-8-carboxylic Acid S. Morris Kupchan and Michael Mokotoff pp 977 - 979; DOI: 10.1021/jm00317a064 |
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A Direct Synthesis of 1-β-D-Arabinofuranosyl-5-fluorocytosine F. Keller, J. E. Bunker, and A. R. Tyrrill pp 979 - 980; DOI: 10.1021/jm00317a065 |
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Terpene Compounds as Drugs. III. Terpenylketoximes Gianfranco Pala, Antonio Mantegani, and Germano Coppi pp 980 - 980; DOI: 10.1021/jm00317a066 |
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Formation of 4-Amino-3,5-di(3-indolylmethyl)-s-triazole from Indole-3-acetonitrile and Hydrazine Robert G. Taborsky pp 980 - 981; DOI: 10.1021/jm00317a067 |
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2-Hydrazino-8-quinolinol and Derivatives Terry Rudolph, F. Przystal, and J. P. Phillips pp 981 - 981; DOI: 10.1021/jm00317a068 |
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3-Aminospirohydantoins Richard A. Wildonger and M. B. Winstead pp 981 - 982; DOI: 10.1021/jm00317a069 |
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Syntheses of Unsymmetric o-Phthalic Acid Diamides Edith G. Díaz de Toranzo and Jorge A. Brieux pp 982 - 983; DOI: 10.1021/jm00317a070 |
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Possible Antifertility Compounds. IV.1 Diphenylnaphtho[1,2-b]- and Diphenylnaphtho[2,1-b]furans S. S. Tiwari and S. C. Srivastava pp 983 - 984; DOI: 10.1021/jm00317a071 |
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Some 2-Aryl-5-nitrobenzimidazole 3-Oxides D. W. Russell pp 984 - 985; DOI: 10.1021/jm00317a072 |
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Flavonoids. V. Thiation of Isoflavones Kenneth H. Dudley, H. Wayne Miller, Robert C. Corley, and Monroe E. Wall pp 985 - 986; DOI: 10.1021/jm00317a073 |
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Synthesis of Potential Antineoplastic Agents. XVIII. Synthesis of New Alkylating Agents Frank D. Popp, Frederick P. Silver, and Adria C. Noble pp 986 - 986; DOI: 10.1021/jm00317a074 |
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Synthesis of Potential Antineoplastic Agents. XIX. Some 5-(ω-Chloroacylamino)quinolines and 4- and 5-(ω-Chloroacylamino)isoquinolines Frederick P. Silver, Frank D. Popp, Adria Catala Casey, D. P. Chakraborty, Ernest Cullen, Warren R. Kirsch, J. E. McCleskey, and Biswajit Sinha pp 986 - 987; DOI: 10.1021/jm00317a075 |
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The Epidemiology of Tropical Diseases. Alfred Burger pp 987 - 987; DOI: 10.1021/jm00317a076 |
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Developmental and Metabolic Control Mechanisms and Neoplasia. Edward J. Modest pp 987 - 988; DOI: 10.1021/jm00317a077 |
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The Story of Health. Alfred Burger pp 988 - 988; DOI: 10.1021/jm00317a078 |
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Advances in Pharmacology. Volume 4. Alfred Burger pp 989 - 989; DOI: 10.1021/jm00317a079 |
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Drug Abuse: Escape to Nowhere. A Guide for Educators. Alfred Burger pp 989 - 989; DOI: 10.1021/jm00317a080 |
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1. Useful Plants of Brazil. 2. A Textbook of Pharmacognosy. Alfred Burger pp 989 - 989; DOI: 10.1021/jm00317a081 |
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Advances in Alicyclic Chemistry. Volume 1. Francis A. Carey pp 989 - 989; DOI: 10.1021/jm00317a082 |
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Russian Drug Index. Alfred Burger pp 989 - 990; DOI: 10.1021/jm00317a083 |
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Index to Reviews, Symposia Volumes and Monographs in Organic Chemistry for the Period 1963-1964. David W. Boykin pp 990 - 990; DOI: 10.1021/jm00317a084 |
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Glass Electrodes for Hydrogen and Other Cations. Principles and Practice. D. R. H. Gourley pp 990 - 990; DOI: 10.1021/jm00317a085 |
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Enzyme and Metabolic Inhibitors. Volumes II and III. Henry A. Lardy pp 990 - 990; DOI: 10.1021/jm00317a086 |
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Quelques Aspects de la Chimie des Médicaments. Alfred Burger pp 990 - 990; DOI: 10.1021/jm00317a087 |
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Analysis of the Structure-Activity Relationship of the Sulfonamide Drugs Using Substituent Constants Toshio Fujita and Corwin Hansch pp 991 - 1000; DOI: 10.1021/jm00318a001 |
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Relationships among Current Quantitative Structure-Activity Models Judith A. Singer and William P. Purcell pp 1000 - 1002; DOI: 10.1021/jm00318a002 |
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The Effect of Piperidinecarboxamide Derivatives on Isolated Cholinesterase Systems. Substituted N1-Benzyl-3-(N,N-diethylcarbamoyl)piperidines James G. Beasley, Samuel T. Christian, W. Ronald Smithfield, and Linda L. Williford pp 1003 - 1005; DOI: 10.1021/jm00318a003 |
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New Norepinephrine-Depleting Agents. β-Hydroxyphenethylguanidine and Related Compounds A. L. Green, R. Fielden, D. C. Bartlett, Mary J. Cozens, R. J. Eden, and D. W. Hills pp 1006 - 1008; DOI: 10.1021/jm00318a004 |
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Tyrosine Hydroxylase Inhibitors. Synthesis and Activity of Substituted Aromatic Amino Acids Walfred S. Saari, June Williams, Susan F. Britcher, Donald E. Wolf, and Frederick A. Kuehl pp 1008 - 1014; DOI: 10.1021/jm00318a005 |
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Aminoalkylindoles with Central Nervous System Activity William J. Welstead, John P. DaVanzo, Grover C. Helsley, Carl D. Lunsford, and C. Roy Taylor pp 1015 - 1021; DOI: 10.1021/jm00318a006 |
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Novel Polycyclic Heterocycles. IV.1 Structure of the Dimer of 5,11-Dihydrodibenz[b,e][1,4]oxazepine. Infrared, Proton Magnetic Resonance, and Mass Spectral Studies Harry L. Yale and Francis Sowinski pp 1022 - 1025; DOI: 10.1021/jm00318a007 |
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The Chemistry and Biological Activity of Derivatives of Strophanthidin S. Morris Kupchan, Michael Mokotoff, Randhir S. Sandhu, and Lowell E. Hokin pp 1025 - 1033; DOI: 10.1021/jm00318a008 |
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Metabolism of (±)-Cotinine-2-14C in the Rat1a,2 Paolo L. Morselli, Helen H. Ong, Edward R. Bowman, and Herbert McKennis pp 1033 - 1036; DOI: 10.1021/jm00318a009 |
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Synthesis and Some Pharmacological Properties of 6-L-Penicillamine-oxytocin Horst Schulz and Vincent Du Vigneaud pp 1037 - 1039; DOI: 10.1021/jm00318a010 |
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The Synthesis, Stereochemistry, and Biology of 16-Hetero and 17-Oxa-D-homo Steroids John S. Baran pp 1039 - 1047; DOI: 10.1021/jm00318a011 |
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Ring-D-Bridged Steroid Analogs. V.1 14α,17α-Etheno-15,16-di(trifluoromethyl)pregna-4,15-diene-3,20-dione and 14α,17α-Ethano-15β,16β-di(trifluoromethyl)pregn-4-ene-3,20- dione2 A. J. Solo and Baldev Singh pp 1048 - 1051; DOI: 10.1021/jm00318a012 |
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Mammalian Antifertility Agents. V. 5,6-Diarylhydronaphthalenones Daniel Lednicer, D. Edward Emmert, Gordon W. Duncan, and Stanley C. Lyster pp 1051 - 1054; DOI: 10.1021/jm00318a013 |
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Stereochemical Aspects of Analgesics. Preparation of 10-Methyl-5-phenyl-5-propionoxy-trans,syn,trans- tetradecahydroacridine Edward E. Smissman and Martin Steinman pp 1054 - 1057; DOI: 10.1021/jm00318a014 |
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Stereochemical Studies on Medicinal Agents. IV.1 Conformational Analysis of Ephedrine Isomers and Related Compounds Philip S. Portoghese pp 1057 - 1063; DOI: 10.1021/jm00318a015 |
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Reaction of Cyclic β-Diketones with 3,4-Dihydroisoquinolines and Related Compounds. Preparation and Anticancer Activity of 2-Substituted 1,3-Cyclohexanediones Max Von Strandtmann, Marvin P. Cohen, and John Shavel pp 1063 - 1065; DOI: 10.1021/jm00318a016 |
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Fluorinated Pyrimidines. XXIX. Syntheses of 2′,3′-Dehydro-5-fluoro-2′-deoxyuridine and 2′,3′-Dideoxy-5-fluorouridine Tasneem A. Khwaja and Charles Heidelberger pp 1066 - 1070; DOI: 10.1021/jm00318a017 |
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Potential Anticancer Agents. III. 2-Phthalimidoaldehydes and Derivatives Jean B. Craig, Claude Piantadosi, J. Logan Irvin, and Shu-Sing Cheng pp 1071 - 1073; DOI: 10.1021/jm00318a018 |
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Imidazolylphosphinamidothionates Henry Tolkmith, Paul B. Budde, Dorsey R. Mussell, and Richard A. Nyquist pp 1074 - 1077; DOI: 10.1021/jm00318a019 |
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A Study of the Synthesis of Barbiturates in Dimethyl Sulfoxide Solvent J. A. Beres, D. E. Pearson, and M. T. Bush pp 1078 - 1080; DOI: 10.1021/jm00318a020 |
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Studies on the Antioxidant Action of Thyroxine and Related Compounds William D. Cash, Harold E. Carlson, Springer W. Cox, Enobong A. Ekong, Jay S. Epstein, and Richard M. Sigel pp 1081 - 1085; DOI: 10.1021/jm00318a021 |
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5,6-Dihydro-4H-1,3,4-thiadiazines. III. Chemistry and Pharmacology of a Series of Basic Derivatives Donald L. Trepanier, Paul E. Krieger, John H. Mennear, and John N. Eble pp 1085 - 1087; DOI: 10.1021/jm00318a022 |
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Synthesis and Amebicidal Activities of Some 1′,2′-Secoemetine Derivatives J. P. Yardley, R. W. Rees, and Herchel Smith pp 1088 - 1091; DOI: 10.1021/jm00318a023 |
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Chemical and Biological Properties of Some Aminomethyl-2-phenylcyclopropane Derivatives. Pharmacological Comparison with Tranylcypromine Uberto M. Teotino, Davide Della Bella, Arnaldo Gandini, and Giancarlo Benelli pp 1091 - 1096; DOI: 10.1021/jm00318a024 |
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The Effects of Bile Acid Derivatives1,2 on Bacterial Permeability and Enzyme Induction Frederick Bernheim and Leon Lack pp 1096 - 1100; DOI: 10.1021/jm00318a025 |
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Irreversible Enzyme Inhibitors. CII. On the Mode of Phenyl Binding of 9-Phenylguanine to Guanine Deaminase and Xanthine Oxidase1-4 B. R. Baker and William F. Wood pp 1101 - 1105; DOI: 10.1021/jm00318a026 |
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Irreversible Enzyme Inhibitors. CIII. 9-(p-Bromoacetamidophenyl)guanine, an Irreversible Inhibitor of Xanthine Oxidase B. R. Baker and William F. Wood pp 1106 - 1109; DOI: 10.1021/jm00318a027 |
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Irreversible Enzyme Inhibitors. CIV. Inhibitors of Thymidine Phosphorylase. VIII. Further Studies on Hydrophobic Bonding with 6-Substituted Uracils B. R. Baker and Waclaw Rzeszotarski pp 1109 - 1113; DOI: 10.1021/jm00318a028 |
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Irreversible Enzyme Inhibitors. CV.1,2 Differential Irreversible Inhibition of Vertebrate Dihydrofolic Reductases by Derivatives of 4,6-Diamino-1,2-dihydro-2,2-dimethyl-1-phenyl-s-triazines Substituted with a Terminal Sulfonyl Fluoride3 B. R. Baker and Gerhardus J. Lourens pp 1113 - 1122; DOI: 10.1021/jm00318a029 |
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Irreversible Enzyme Inhibitors. CVI.1 Proteolytic Enzymes. I. Bulk Tolerances in Trypsin-Inhibitor Complexes2 B. R. Baker and Edward H. Erickson pp 1123 - 1128; DOI: 10.1021/jm00318a030 |
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Irreversible Enzyme Inhibitors. CVII.1 Proteolytic Enzymes. II.2 Bulk Tolerance within Chymotrypsin-Inhibitor Complexes B. R. Baker and Jeffrey A. Hurlbut pp 1129 - 1133; DOI: 10.1021/jm00318a031 |
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Irreversible Enzyme Inhibitors. CVIII.1,2 6-(p-Chloroacetylanilinomethyl)-5-(p-chlorophenyl)-2, 4-diaminopyrimidine, an Active-Site-Directed Irreversible Inhibitor of Dihydrofolic Reductase B. R. Baker, Ping Cheong Huang, and Alfonso L. Pogolotti pp 1134 - 1138; DOI: 10.1021/jm00318a032 |
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2,2′-Hydrazobis(5-nitrothiazoles) and Analogs, a New Type of Antiprotozoal Agents Moshe Avramoff, Saul Adler, and Ann Foner pp 1138 - 1143; DOI: 10.1021/jm00318a033 |
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Synthesis and Biological Screening of Aminotropone Derivatives E. Sianesi, P. Da Re, M. J. Magistretti, and I. Setnikar pp 1144 - 1148; DOI: 10.1021/jm00318a034 |
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A New Antibiotic. Furanomycin, an Isoleucine Antagonist Ken Katagiri, Kazuo Tori, Yasuo Kimura, Tadashi Yoshida, Tohru Nagasaki, and Hitoshi Minato pp 1149 - 1154; DOI: 10.1021/jm00318a035 |
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Synthesis and Evaluation of the Local Anesthetic Activity of a Series of 2-Alkoxy-4-(ω-alkylaminoacylamino)benzoic Acid Esters George Tsatsas, Demetrios Kontonassios, and Constantine Sandris pp 1154 - 1157; DOI: 10.1021/jm00318a036 |
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Synthesis and Enzymological Activity of Some Pyridoxine Analogs Paul Melius and David L. Marshall pp 1157 - 1158; DOI: 10.1021/jm00318a037 |
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Metabolism of 5-(3-Pyridyl)tetrazole S. K. Figdor and M. Schach von Wittenau pp 1158 - 1159; DOI: 10.1021/jm00318a038 |
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1-(1-Indanyl)- and 1-(1-Tetralyl)imidazole-5-carboxylate Esters, a Novel Type of Antifungal Agents Erik F. Godefroi, Jan Van Cutsem, Cyriel A. M. Van der Eycken, and Paul A. J. Janssen pp 1160 - 1161; DOI: 10.1021/jm00318a039 |
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Lincomycin. VII. 4′-Depropyl-4′-ethoxylincomycins Barney J. Magerlein pp 1161 - 1163; DOI: 10.1021/jm00318a040 |
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Bis(pyrimidine nucleoside) Phosphates John A. Montgomery and H. Jeanette Thomas pp 1163 - 1165; DOI: 10.1021/jm00318a041 |
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3′-Deoxynucleosides. V. 3′-Deoxy-2-fluoroadenosine Mary J. Dickinson, Frederick W. Holly, Edward Walton, and Morris Zimmerman pp 1165 - 1166; DOI: 10.1021/jm00318a042 |
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Organic Disulfides and Related Substances. XXIV. Unsymmetrical n-Decylaminoethyl Disulfides as Antiradiation Drugs Lamar Field, H. K. Kim, and Michael Bellas pp 1166 - 1167; DOI: 10.1021/jm00318a043 |
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Trifluoromethyl Thiolsulfonates and Their Reactions with Mercaptans and Amines J. P. Weidner and S. S. Block pp 1167 - 1170; DOI: 10.1021/jm00318a044 |
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The Effect of Some Disulfides and Thiols on the Carbohydrate Metabolism of Ehrlich Ascites Tumor D. R. Grassetti, J. F. Murray, M. E. Brokke, and A. D. Gutman pp 1170 - 1172; DOI: 10.1021/jm00318a045 |
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Amides of N-Acylcysteines as Mucolytic Agents Tellis A. Martin, David H. Causey, A. Leonard Sheffner, Allan G. Wheeler, and John R. Corrigan pp 1172 - 1176; DOI: 10.1021/jm00318a046 |
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Synthesis and Reactions of Some Pyrimidylethyl Isocyanates C. E. Morreal, J. H. Hall, and K. Eskins pp 1176 - 1178; DOI: 10.1021/jm00318a047 |
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Substituted 1-Benzyl-3-(N,N-diethylcarbamoyl)-piperidine Cholinesterase Inhibitors. Relationships between Molecular Constitution, pKa' Values, and Partition Coefficients Ronald P. Quintana and W. Ronald Smithfield pp 1178 - 1180; DOI: 10.1021/jm00318a048 |
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Acetylenic Carbamates. II. Reactions of 1,1-Diaryl-2-propynyl Carbamates with Acids and Bases Robert D. Dillard, Donald R. Cassady, and Nelson R. Easton pp 1180 - 1182; DOI: 10.1021/jm00318a049 |
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Some 2,3,6,8-Tetrasubstituted Quinazolone Hydrazides as Monoamine Oxidase Inhibitors Surendra S. Parmar and R. C. Arora pp 1182 - 1183; DOI: 10.1021/jm00318a050 |
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2-Thio-1,3,4,6,7,11b-hexahydro-9,10-dimethoxy-2H-benzo[a]quinolizines M. R. Harnden and J H. Short pp 1183 - 1184; DOI: 10.1021/jm00318a051 |
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Some 2,6-Methanonaphth[1,2-d]azocines Robert L. Perry and N. F. Albertson pp 1184 - 1186; DOI: 10.1021/jm00318a052 |
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Effect of Organic Compounds on Reproductive Processes. VII. Bis-N,N′-carbamoylaziridines W. A. Skinner, M. Cory, and J. I. DeGraw pp 1186 - 1188; DOI: 10.1021/jm00318a053 |
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A Synthesis of 11β-Hydroxyestrone and Related 16- and 17-Hydroxyestratrienes John S. Baran pp 1188 - 1190; DOI: 10.1021/jm00318a054 |
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Insect Sex Attractants. VII. 5,9-Tridecadien-1-ol Acetates David Warthen and Martin Jacobson pp 1190 - 1191; DOI: 10.1021/jm00318a055 |
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Some Semicarbazones and Thiosemicarbazones Abelardo P. Martinez and William W. Lee pp 1192 - 1192; DOI: 10.1021/jm00318a056 |
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Trifluoromethylbenzaldoximes Charles F. Barfknecht and Tim R. Westby pp 1192 - 1193; DOI: 10.1021/jm00318a057 |
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Anticancer Agents. John M. Venditti pp 1193 - 1194; DOI: 10.1021/jm00318a058 |
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Progress in Drug Research. Volume 10. Alfred Burger pp 1194 - 1194; DOI: 10.1021/jm00318a059 |
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Topics in Medicinal Chemistry. Volume 1. Alfred Burger pp 1194 - 1195; DOI: 10.1021/jm00318a060 |
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2-Thio-1,3,4,6,7,11b-hexahydro-9,10-dimethoxy- 2H-benzo[a]quinolizines M. R. Harnden and J. H. Short pp 1195 - 1195; DOI: 10.1021/jm00318a061 |
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Dilemmas in Drug Therapy. Alfred Burger pp 1195 - 1195; DOI: 10.1021/jm00318a062 |
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Psychotropic Drugs and Related Compounds. Alfred Burger pp 1195 - 1195; DOI: 10.1021/jm00318a063 |
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Problemès Actuels de Biochimie Appliqueé. Alfred Burger pp 1195 - 1196; DOI: 10.1021/jm00318a064 |
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Design of Active-Site-Directed Irreversible Enzyme Inhibitors. Alfred Burger pp 1196 - 1196; DOI: 10.1021/jm00318a065 |
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Principles of Scientific and Technical Writing. Alfred Burger pp 1196 - 1196; DOI: 10.1021/jm00318a066 |
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Organic Photochemistry. Volume 1. Francis A. Carey pp 1196 - 1196; DOI: 10.1021/jm00318a067 |
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Problems in Laboratory Evaluation of Antianginal Agents. Alfred Burger pp 1197 - 1197; DOI: 10.1021/jm00318a068 |
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Additions and Corrections - Monothiophenyl Malonate. John C. Howard, Michael C. Lin, Patricia Matthews, and Sam A. Singal pp 1197 - 1197; DOI: 10.1021/jm00318a069 |
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Additions and Corrections - 3-Substituted 2-Thiohydrouracils. Synthesis and Antitubercular and Antineoplastic Activities. Arthur C. Glasser, and Richard M. Doughty pp 1197 - 1197; DOI: 10.1021/jm00318a600 |
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Additions and Corrections - 3-Pheylcinnolines. I. Some Reactions and Derivatives of 3-Phenylcinnoline-4-carboxylic Acids. Harman S. Lowrie pp 1197 - 1197; DOI: 10.1021/jm00318a601 |
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Additions and Corrections - Pteridinecarboxamide Diuretics. I. Reaction of 4,6-Diamino-5-nitrosopyrimidines with Substituted Malonamides. T. S. Osdene, Arthur A. Santilli, Lee E. McCardle, and Marvin E. Rosenthale pp 1197 - 1197; DOI: 10.1021/jm00318a602 |
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Additions and Corrections - Benzo(b)thiopene Derivatives. Synthesis and Pharmacology. N. B. Chapman, K. Clarke, and B. Iddon pp 1197 - 1197; DOI: 10.1021/jm00318a603 |
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Additions and Corrections - Synthetic Bradykinin Analogs. Ernest Nicolaides, and Marilyn Lipnik pp 1197 - 1197; DOI: 10.1021/jm00318a604 |
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Additions and Corrections - 16-Aza Steroids. R. W. Kierstead, A. Farsone, and A. Boris pp 1197 - 1197; DOI: 10.1021/jm00318a605 |
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Additions and Corrections - Substituted 2,3-Dihydro-4(1H)-quinazolinones. A New Class of Inhibitors of Cell Multiplication. Harry L. Yale, and Marion Kalkstein pp 1197 - 1197; DOI: 10.1021/jm00318a606 |
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Additions and Corrections - New Psychotropic Agents. VIII. Analogs of Amitriptyline Containing the Normeperidine Group. M. A. Davis, F. Herr, R. A. Thomas, and Marie-Paule Charest pp 1197 - 1197; DOI: 10.1021/jm00318a607 |
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Additions and Corrections - Potential Carcinostatic Agents. I. Derivatives and Analogs of 1-(2-Hydroxyethyl)-3-(4-tolyl)urea. Harold G. Nelson, Frederic J. Shelton, and William H. Wetzel pp 1197 - 1197; DOI: 10.1021/jm00318a608 |